Anastrozole, estrogen buster

 KNOWLEDGE    |      2023-03-28

Mabasi a Estrogen


Anastrozole ndi mankhwala amphamvu oletsa akazi omwe ali mu aromatase inhibitor, omwe ndi mankhwala otchuka pakati pa omanga thupi.


Anastrozole amagwiritsidwa ntchito ndi ogwiritsa ntchito ambiri a steroid panthawi yozungulira kuti athetsere zomwe zimachitika. Ma steroid ambiri aromatize ndipo amayambitsa zotsatira za estrogen, zomwe anastrozole ndi njira yabwino yothetsera. Zimachepetsa testosterone m'thupi ndi 80 peresenti. Ichi ndi phindu lamtengo wapatali kwa ogwiritsa ntchito steroid, komanso kulimbikitsa kupanga kwa hormone ya luteinizing ndi follicle stimulating hormone.


Kwa ogwiritsira ntchito steroid, anastrozole amalepheretsa zotsatira za mankhwala a inofemale reaction. Chifukwa ma steroid ambiri amanunkhira m'thupi ndipo amasandulika kukhala estrogen, zomwe zingayambitse zotsatira zoyipa. Pa ma steroids, milingo ya estrogen mwa ogwiritsa ntchito imakwera pafupifupi kuwirikiza kasanu ndi kawiri kuposa omwe sagwiritsa ntchito, zomwe zimapangitsa kuti madzi asungidwe kwambiri komanso nsonga ya mabere ectosis ikasiyidwa. Aromatase inhibitors monga anastrozole ndiwothandiza kwambiri pakuwongolera oecytosis, pomwe ma modulators osankhidwa ogonana ogonana monga tamoxifen sagwira ntchito kwambiri kuposa Mlingo wa 0.5-MG ndiofala kwambiri kwa ogwiritsa ntchito ma steroid. Ndi anthu ochepa okha amene adzafunika gigabyte yoposa imodzi, ndipo nthawi zambiri imakhala yokwanira. Koma othamanga asanayambe mpikisano angaone kuti ndizothandiza kutenga 0.5MG ya anastrozole tsiku kwa masiku 10 mpaka 14 kuti akhwime minofu.


Zimalimbikitsidwanso kuti muwonjezere anastrozole mu PCT kuchira, zomwe zingathe kusunga chiŵerengero cha estrogen ku testosterone mkati mwamtundu wamba. Kuphatikiza apo, anastrozole imawonjezera kuchuluka kwa timadzi ta luteinizing ndi follicle-stimulating hormone, ndipo testosterone yoponderezedwa imatha kuchira msanga mwachangu.