Anastrozole, busteri ya estrogene

 KNOWLEDGE    |      2023-03-28

Estrogen busters


Anastrozole ni imiti ikomeye igabanya ubukana bwa aromatase inhibitor, ikaba ari imiti izwi cyane mu bubaka umubiri.


Anastrozole ikoreshwa nabakoresha steroid batabarika mugihe cyo kuzenguruka kugirango bahagarike reaction. Steroide nyinshi zihumura kandi zigatera ingaruka za estrogene, anastrozole nigisubizo cyiza kuri. Mu byukuri igabanya urugero rwa testosterone mu mubiri 80%. Iyi ninyungu zingirakamaro kubakoresha steroid, kimwe no gushishikariza gukora imisemburo ya luteinizing na follicle itera imisemburo


Kubakoresha steroid, anastrozole ibuza ingaruka ziterwa nibiyobyabwenge byabagore. Kuberako steroide nyinshi ihumura mumubiri igahinduka estrogene, ishobora gutera ingaruka. Kuri steroyide, urugero rwa estrogene mubakoresha irazamuka kugera ku kigereranyo cyikubye inshuro zirindwi ugereranije n’abatayikoresha, bigatuma ububiko bw’amazi bukabije hamwe n’amabere ya ectose iyo bidasuzumwe. Inzitizi ya Aromatase nka anastrozole ningirakamaro cyane mugucunga oecytose, mugihe modulator zo mu bwoko bwa hormone zo mu mibonano mpuzabitsina nka tamoxifen zidakora neza cyane kuruta dosiye ya 0.5-MG ikunze kugaragara kubakoresha steroid. Abantu bake cyane bazakenera gigabyte zirenze imwe, kandi mubihe byinshi birahagije rwose. Ariko abakinnyi babanjirije amarushanwa bashobora gusanga ari byiza gufata 0.5MG ya anastrozole kumunsi muminsi 10 kugeza 14 kugirango bakomere imitsi


Birasabwa kandi kongeramo anastrozole mugusubirana kwa PCT, ishobora kugumana igipimo cya estrogene na testosterone murwego rusanzwe. Byongeye kandi, anastrozole yongerera urwego imisemburo ya luteinizing na hormone itera imisemburo, kandi testosterone ihagaritswe irashobora gukira kurwego rusanzwe vuba.