Anastrozole, inonzi estrogen buster

 KNOWLEDGE    |      2023-03-28

Estrogen busters


Anastrozole mushonga une simba wevakadzi uri we aromatase inhibitor, inova inodhaka inorwisa vakadzi pakati pevanovaka muviri.


Anastrozole inoshandiswa nevakawanda vashandisi ve steroid panguva yekutenderera kudzvinyirira maitiro ekuita. Mazhinji steroid aromatize uye anokonzera estrogen mhedzisiro, iyo anastrozole mhinduro yakanaka kune. Iyo inoderedza mazinga e testosterone mumuviri ne80 muzana. Ichi chibatsiro chakakosha kune vashandisi ve steroid, pamwe nekukurudzira kugadzirwa kwe luteinizing hormone uye follicle stimulating hormone.


Kune vashandisi ve steroid, anastrozole inhibits mhedzisiro yemushonga inofemale reaction. Nekuti akawanda steroid anonhuhwirira mumuviri uye anoshandurwa kuita estrogen, izvo zvinogona kukonzera mhedzisiro. Pamasteroids, mazinga eesrogen muvashandisi anokwira kusvika paavhareji yakapetwa kanomwe kupfuura yevasiri vashandisi, zvichikonzera kuchengetwa kwemvura kwakanyanya uye mazamu tip ectosis kana isina kubatwa. Aromatase inhibitors akadai seanastrozole ndiyo inonyanya kushanda pakudzora oecytosis, nepo sarudzo dzepabonde dzepabonde modulators dzakadai setamoxifen dzisinganyanyi kushanda pane madosi e0.5-MG akajairika kune vashandisi vesteroid. Vashoma vanhu vanozoda anopfuura gigabyte imwe, uye kazhinji inokwana zvakakwana. Asi vatambi vasati vakwikwidza vanogona kuona zvichibatsira kutora 0.5MG yeanastrozole pazuva kwemazuva gumi kusvika gumi nemana kuomesa tsandanyama.


Inokurudzirwawo kuwedzera anastrozole muPCT kupora, iyo inogona kuchengetedza chiyero cheesrogen kune testosterone mukati mehutano hwemazuva ose. Mukuwedzera, anastrozole inowedzera mazinga e luteinizing hormone uye follicle-stimulating hormone, uye yakadzvinyirirwa endo native testosterone inogona kupora kusvika kune yakajairika nhanho nekukurumidza.